Xyzal (levocetirizine) dosing, indications, interactions, adverse effects, and more (2024)

  • acetaminophen/phenyltoloxamine

    levocetirizine and acetaminophen/phenyltoloxamine both increase sedation. Use Caution/Monitor.

  • acrivastine

    acrivastine and levocetirizine both increase sedation. Use Caution/Monitor.

  • alprazolam

    levocetirizine and alprazolam both increase sedation. Use Caution/Monitor.

  • amifampridine

    levocetirizine increases toxicity of amifampridine by Other (see comment). Modify Therapy/Monitor Closely. Comment: Amifampridine can cause seizures. Coadministration with drugs that lower seizure threshold may increase this risk.

  • amisulpride

    amisulpride and levocetirizine both increase sedation. Use Caution/Monitor.

  • amitriptyline

    levocetirizine and amitriptyline both increase sedation. Use Caution/Monitor.

  • amobarbital

    levocetirizine and amobarbital both increase sedation. Use Caution/Monitor.

  • amoxapine

    levocetirizine and amoxapine both increase sedation. Use Caution/Monitor.

  • aripiprazole

    levocetirizine and aripiprazole both increase sedation. Use Caution/Monitor.

  • asenapine

    asenapine and levocetirizine both increase sedation. Use Caution/Monitor.

  • asenapine transdermal

    asenapine transdermal and levocetirizine both increase sedation. Use Caution/Monitor.

  • avapritinib

    avapritinib and levocetirizine both increase sedation. Use Caution/Monitor.

  • baclofen

    levocetirizine and baclofen both increase sedation. Use Caution/Monitor.

  • benzhydrocodone/acetaminophen

    benzhydrocodone/acetaminophen and levocetirizine both increase sedation. Use Caution/Monitor.

  • brexanolone

    levocetirizine and brexanolone both increase sedation. Use Caution/Monitor.

  • brexpiprazole

    brexpiprazole and levocetirizine both increase sedation. Use Caution/Monitor.

  • brimonidine

    brimonidine and levocetirizine both increase sedation. Use Caution/Monitor.

  • brivaracetam

    brivaracetam and levocetirizine both increase sedation. Use Caution/Monitor.

  • brompheniramine

    levocetirizine and brompheniramine both increase sedation. Use Caution/Monitor.

  • buprenorphine subdermal implant

    buprenorphine subdermal implant and levocetirizine both increase sedation. Use Caution/Monitor.

  • buprenorphine transdermal

    buprenorphine transdermal and levocetirizine both increase sedation. Use Caution/Monitor.

  • buprenorphine, long-acting injection

    buprenorphine, long-acting injection and levocetirizine both increase sedation. Use Caution/Monitor.

  • butabarbital

    levocetirizine and butabarbital both increase sedation. Use Caution/Monitor.

  • butalbital

    levocetirizine and butalbital both increase sedation. Use Caution/Monitor.

  • butorphanol

    levocetirizine and butorphanol both increase sedation. Use Caution/Monitor.

  • carbinoxamine

    levocetirizine and carbinoxamine both increase sedation. Use Caution/Monitor.

  • cariprazine

    cariprazine and levocetirizine both increase sedation. Use Caution/Monitor.

  • carisoprodol

    levocetirizine and carisoprodol both increase sedation. Use Caution/Monitor.

  • cenobamate

    levocetirizine and cenobamate both increase sedation. Use Caution/Monitor.

  • cetirizine

    levocetirizine and cetirizine both increase sedation. Use Caution/Monitor.

  • chlordiazepoxide

    levocetirizine and chlordiazepoxide both increase sedation. Use Caution/Monitor.

  • chlorpheniramine

    levocetirizine and chlorpheniramine both increase sedation. Use Caution/Monitor.

  • chlorpromazine

    levocetirizine and chlorpromazine both increase sedation. Use Caution/Monitor.

  • chlorzoxazone

    levocetirizine and chlorzoxazone both increase sedation. Use Caution/Monitor.

  • clemastine

    levocetirizine and clemastine both increase sedation. Use Caution/Monitor.

  • clobazam

    levocetirizine, clobazam. Other (see comment). Use Caution/Monitor. Comment: Concomitant administration can increase the potential for CNS effects (e.g., increased sedation or respiratory depression).levocetirizine and clobazam both increase sedation. Use Caution/Monitor.

  • clomipramine

    levocetirizine and clomipramine both increase sedation. Use Caution/Monitor.

  • clonazepam

    levocetirizine and clonazepam both increase sedation. Use Caution/Monitor.

  • clonidine

    levocetirizine and clonidine both increase sedation. Use Caution/Monitor.

  • clorazepate

    levocetirizine and clorazepate both increase sedation. Use Caution/Monitor.

  • clozapine

    levocetirizine and clozapine both increase sedation. Use Caution/Monitor.

  • cyclobenzaprine

    levocetirizine and cyclobenzaprine both increase sedation. Use Caution/Monitor.

  • cyproheptadine

    levocetirizine and cyproheptadine both increase sedation. Use Caution/Monitor.

  • dantrolene

    levocetirizine and dantrolene both increase sedation. Use Caution/Monitor.

  • daridorexant

    levocetirizine and daridorexant both increase sedation. Modify Therapy/Monitor Closely. Coadministration increases risk of CNS depression, which can lead to additive impairment of psychom*otor performance and cause daytime impairment.

  • desflurane

    levocetirizine and desflurane both increase sedation. Use Caution/Monitor.

  • desipramine

    levocetirizine and desipramine both increase sedation. Use Caution/Monitor.

  • desloratadine

    desloratadine and levocetirizine both increase sedation. Use Caution/Monitor.

  • deutetrabenazine

    levocetirizine and deutetrabenazine both increase sedation. Use Caution/Monitor.

  • dexbrompheniramine

    levocetirizine and dexbrompheniramine both increase sedation. Use Caution/Monitor.

  • dexchlorpheniramine

    levocetirizine and dexchlorpheniramine both increase sedation. Use Caution/Monitor.

  • diazepam

    levocetirizine and diazepam both increase sedation. Use Caution/Monitor.

  • diazepam intranasal

    diazepam intranasal, levocetirizine.Either increases effects of the other by pharmacodynamic synergism. Use Caution/Monitor. Coadministration may potentiate the CNS-depressant effects of each drug.

  • difenoxin hcl

    levocetirizine and difenoxin hcl both increase sedation. Use Caution/Monitor.

  • dimenhydrinate

    levocetirizine and dimenhydrinate both increase sedation. Use Caution/Monitor.

  • diphenhydramine

    levocetirizine and diphenhydramine both increase sedation. Use Caution/Monitor.

  • diphenoxylate hcl

    levocetirizine and diphenoxylate hcl both increase sedation. Use Caution/Monitor.

  • donepezil transdermal

    donepezil transdermal, levocetirizine.Either decreases effects of the other by pharmacodynamic antagonism. Use Caution/Monitor.

  • doxepin

    levocetirizine and doxepin both increase sedation. Use Caution/Monitor.

  • doxylamine

    levocetirizine and doxylamine both increase sedation. Use Caution/Monitor.

  • droperidol

    levocetirizine and droperidol both increase sedation. Use Caution/Monitor.

  • efavirenz

    levocetirizine and efavirenz both increase sedation. Use Caution/Monitor.

  • entacapone

    levocetirizine and entacapone both increase sedation. Use Caution/Monitor.

  • esketamine intranasal

    esketamine intranasal, levocetirizine.Either increases toxicity of the other by sedation. Modify Therapy/Monitor Closely.

  • estazolam

    levocetirizine and estazolam both increase sedation. Use Caution/Monitor.

  • eszopiclone

    levocetirizine and eszopiclone both increase sedation. Use Caution/Monitor.

  • ethanol

    levocetirizine and ethanol both increase sedation. Use Caution/Monitor.

  • ethosuximide

    levocetirizine and ethosuximide both increase sedation. Use Caution/Monitor.

  • ethotoin

    levocetirizine and ethotoin both increase sedation. Use Caution/Monitor.

  • felbamate

    levocetirizine and felbamate both increase sedation. Use Caution/Monitor.

  • fenfluramine

    levocetirizine and fenfluramine both increase sedation. Use Caution/Monitor.

  • fentanyl

    fentanyl and levocetirizine both increase sedation. Use Caution/Monitor.

  • fentanyl intranasal

    fentanyl intranasal and levocetirizine both increase sedation. Use Caution/Monitor.

  • fentanyl iontophoretic transdermal system

    fentanyl iontophoretic transdermal system and levocetirizine both increase sedation. Use Caution/Monitor.

  • fentanyl transdermal

    fentanyl transdermal and levocetirizine both increase sedation. Use Caution/Monitor.

  • fentanyl transmucosal

    fentanyl transmucosal and levocetirizine both increase sedation. Use Caution/Monitor.

  • fexofenadine

    levocetirizine and fexofenadine both increase sedation. Use Caution/Monitor.

  • flibanserin

    levocetirizine and flibanserin both increase sedation. Use Caution/Monitor.

  • fluphenazine

    levocetirizine and fluphenazine both increase sedation. Use Caution/Monitor.

  • flurazepam

    levocetirizine and flurazepam both increase sedation. Use Caution/Monitor.

  • gabapentin

    gabapentin, levocetirizine.Either increases effects of the other by pharmacodynamic synergism. Modify Therapy/Monitor Closely. Coadministration of CNS depressants can result in serious, life-threatening, and fatal respiratory depression. Use lowest dose possible and monitor for respiratory depression and sedation.levocetirizine and gabapentin both increase sedation. Use Caution/Monitor.

  • gabapentin enacarbil

    gabapentin enacarbil, levocetirizine.Either increases effects of the other by pharmacodynamic synergism. Modify Therapy/Monitor Closely. Coadministration of CNS depressants can result in serious, life-threatening, and fatal respiratory depression. Use lowest dose possible and monitor for respiratory depression and sedation.

  • ganaxolone

    levocetirizine and ganaxolone both increase sedation. Use Caution/Monitor.

  • guanfacine

    levocetirizine and guanfacine both increase sedation. Use Caution/Monitor.

  • haloperidol

    levocetirizine and haloperidol both increase sedation. Use Caution/Monitor.

  • hyaluronidase

    levocetirizine decreases effects of hyaluronidase by Other (see comment). Use Caution/Monitor. Comment: Antihistamines, when given in large systemic doses, may render tissues partially resistant to the action of hyaluronidase. Patients may require larger amounts of hyaluronidase for equivalent dispersing effect. .

  • hydroxyzine

    levocetirizine and hydroxyzine both increase sedation. Use Caution/Monitor.

  • iloperidone

    levocetirizine and iloperidone both increase sedation. Use Caution/Monitor.

  • imipramine

    levocetirizine and imipramine both increase sedation. Use Caution/Monitor.

  • isoflurane

    levocetirizine and isoflurane both increase sedation. Use Caution/Monitor.

  • ketamine

    levocetirizine and ketamine both increase sedation. Use Caution/Monitor.

  • ketotifen, drug-eluting contact lens

    levocetirizine and ketotifen, drug-eluting contact lens both increase sedation. Use Caution/Monitor.

  • lamotrigine

    levocetirizine and lamotrigine both increase sedation. Use Caution/Monitor.

  • lasmiditan

    levocetirizine and lasmiditan both increase sedation. Use Caution/Monitor.

  • lemborexant

    levocetirizine and lemborexant both increase sedation. Use Caution/Monitor.

  • levetiracetam

    levetiracetam and levocetirizine both increase sedation. Use Caution/Monitor.levocetirizine and levetiracetam both increase sedation. Use Caution/Monitor.

  • levorphanol

    levocetirizine and levorphanol both increase sedation. Use Caution/Monitor.

  • loratadine

    levocetirizine and loratadine both increase sedation. Use Caution/Monitor.loratadine and levocetirizine both increase sedation. Use Caution/Monitor.

  • lorazepam

    levocetirizine and lorazepam both increase sedation. Use Caution/Monitor.

  • loxapine

    levocetirizine and loxapine both increase sedation. Use Caution/Monitor.

  • lumateperone

    levocetirizine and lumateperone both increase sedation. Use Caution/Monitor.lumateperone and levocetirizine both increase sedation. Use Caution/Monitor.

  • lurasidone

    lurasidone, levocetirizine.Either increases toxicity of the other by Other (see comment). Use Caution/Monitor. Comment: Potential for increased CNS depressant effects when used concurrently; monitor for increased adverse effects and toxicity.levocetirizine and lurasidone both increase sedation. Use Caution/Monitor.

  • maprotiline

    levocetirizine and maprotiline both increase sedation. Use Caution/Monitor.

  • meclizine

    levocetirizine and meclizine both increase sedation. Use Caution/Monitor.

  • meperidine

    levocetirizine and meperidine both increase sedation. Use Caution/Monitor.

  • meprobamate

    levocetirizine and meprobamate both increase sedation. Use Caution/Monitor.

  • metaxalone

    levocetirizine and metaxalone both increase sedation. Use Caution/Monitor.

  • methocarbamol

    levocetirizine and methocarbamol both increase sedation. Use Caution/Monitor.

  • methohexital

    methohexital and levocetirizine both increase sedation. Use Caution/Monitor.levocetirizine and methohexital both increase sedation. Use Caution/Monitor.

  • methsuximide

    levocetirizine and methsuximide both increase sedation. Use Caution/Monitor.

  • midazolam

    levocetirizine and midazolam both increase sedation. Use Caution/Monitor.

  • midazolam intranasal

    midazolam intranasal, levocetirizine.Either increases toxicity of the other by pharmacodynamic synergism. Modify Therapy/Monitor Closely. Concomitant use of barbiturates, alcohol, or other CNS depressants may increase the risk of hypoventilation, airway obstruction, desaturation, or apnea and may contribute to profound and/or prolonged drug effect.

  • mirtazapine

    levocetirizine and mirtazapine both increase sedation. Use Caution/Monitor.

  • molindone

    levocetirizine and molindone both increase sedation. Use Caution/Monitor.

  • nalbuphine

    levocetirizine and nalbuphine both increase sedation. Use Caution/Monitor.

  • nitrous oxide

    levocetirizine and nitrous oxide both increase sedation. Use Caution/Monitor.

  • nortriptyline

    levocetirizine and nortriptyline both increase sedation. Use Caution/Monitor.

  • olanzapine

    levocetirizine and olanzapine both increase sedation. Use Caution/Monitor.

  • olanzapine/samidorphan

    levocetirizine and olanzapine/samidorphan both increase sedation. Use Caution/Monitor.

  • oliceridine

    levocetirizine and oliceridine both increase sedation. Use Caution/Monitor.

  • opicapone

    levocetirizine and opicapone both increase sedation. Use Caution/Monitor.

  • opium tincture

    levocetirizine and opium tincture both increase sedation. Use Caution/Monitor.

  • orphenadrine

    levocetirizine and orphenadrine both increase sedation. Use Caution/Monitor.

  • oxazepam

    levocetirizine and oxazepam both increase sedation. Use Caution/Monitor.

  • paliperidone

    levocetirizine and paliperidone both increase sedation. Use Caution/Monitor.

  • pentazocine

    levocetirizine and pentazocine both increase sedation. Use Caution/Monitor.

  • pentobarbital

    levocetirizine and pentobarbital both increase sedation. Use Caution/Monitor.

  • perampanel

    levocetirizine and perampanel both increase sedation. Use Caution/Monitor.

  • perphenazine

    levocetirizine and perphenazine both increase sedation. Use Caution/Monitor.

  • phenelzine

    phenelzine increases effects of levocetirizine by Other (see comment). Modify Therapy/Monitor Closely. Comment: Coadministration of phenelzine and antihistamines may result in additive CNS depressant effects. MAO inhibitors also prolong and intensify anticholinergic effects of antihistamines. .

  • pheniramine

    levocetirizine and pheniramine both increase sedation. Use Caution/Monitor.

  • phenobarbital

    levocetirizine and phenobarbital both increase sedation. Use Caution/Monitor.

  • pimozide

    levocetirizine and pimozide both increase sedation. Use Caution/Monitor.

  • pomalidomide

    levocetirizine and pomalidomide both increase sedation. Use Caution/Monitor.

  • pregabalin

    pregabalin, levocetirizine.Either increases effects of the other by pharmacodynamic synergism. Modify Therapy/Monitor Closely. Coadministration of CNS depressants can result in serious, life-threatening, and fatal respiratory depression. Use lowest dose possible and monitor for respiratory depression and sedation.levocetirizine and pregabalin both increase sedation. Use Caution/Monitor.

  • primidone

    levocetirizine and primidone both increase sedation. Use Caution/Monitor.

  • prochlorperazine

    levocetirizine and prochlorperazine both increase sedation. Use Caution/Monitor.

  • promethazine

    levocetirizine and promethazine both increase sedation. Use Caution/Monitor.

  • propofol

    levocetirizine and propofol both increase sedation. Use Caution/Monitor.

  • protriptyline

    levocetirizine and protriptyline both increase sedation. Use Caution/Monitor.

  • pyrilamine

    levocetirizine and pyrilamine both increase sedation. Use Caution/Monitor.

  • quazepam

    levocetirizine and quazepam both increase sedation. Use Caution/Monitor.

  • quetiapine

    levocetirizine and quetiapine both increase sedation. Use Caution/Monitor.

  • ramelteon

    levocetirizine and ramelteon both increase sedation. Use Caution/Monitor.

  • remimazolam

    levocetirizine and remimazolam both increase sedation. Use Caution/Monitor.

  • reserpine

    levocetirizine and reserpine both increase sedation. Use Caution/Monitor.

  • risperidone

    levocetirizine and risperidone both increase sedation. Use Caution/Monitor.

  • ritonavir

    ritonavir increases levels of levocetirizine by decreasing metabolism. Use Caution/Monitor.

  • scopolamine

    levocetirizine and scopolamine both increase sedation. Use Caution/Monitor.

  • sevoflurane

    levocetirizine and sevoflurane both increase sedation. Use Caution/Monitor.

  • sodium oxybate

    levocetirizine and sodium oxybate both increase sedation. Use Caution/Monitor.

  • stiripentol

    stiripentol, levocetirizine.Either increases effects of the other by sedation. Use Caution/Monitor. Concomitant use stiripentol with other CNS depressants, including alcohol, may increase the risk of sedation and somnolence.

  • sufentanil

    levocetirizine and sufentanil both increase sedation. Use Caution/Monitor.

  • sufentanil SL

    levocetirizine and sufentanil SL both increase sedation. Use Caution/Monitor.

  • suvorexant

    levocetirizine and suvorexant both increase sedation. Use Caution/Monitor.

  • tapentadol

    levocetirizine and tapentadol both increase sedation. Use Caution/Monitor.

  • tasimelteon

    levocetirizine and tasimelteon both increase sedation. Use Caution/Monitor.

  • temazepam

    levocetirizine and temazepam both increase sedation. Use Caution/Monitor.

  • tetrabenazine

    levocetirizine and tetrabenazine both increase sedation. Use Caution/Monitor.

  • thioridazine

    levocetirizine and thioridazine both increase sedation. Use Caution/Monitor.

  • thiothixene

    levocetirizine and thiothixene both increase sedation. Use Caution/Monitor.

  • tiagabine

    levocetirizine and tiagabine both increase sedation. Use Caution/Monitor.

  • tizanidine

    levocetirizine and tizanidine both increase sedation. Use Caution/Monitor.

  • tolcapone

    levocetirizine and tolcapone both increase sedation. Use Caution/Monitor.

  • topiramate

    levocetirizine and topiramate both increase sedation. Use Caution/Monitor.

  • trazodone

    levocetirizine and trazodone both increase sedation. Use Caution/Monitor.

  • trifluoperazine

    levocetirizine and trifluoperazine both increase sedation. Use Caution/Monitor.

  • triprolidine

    levocetirizine and triprolidine both increase sedation. Use Caution/Monitor.

  • valproic acid

    levocetirizine and valproic acid both increase sedation. Use Caution/Monitor.

  • vigabatrin

    levocetirizine and vigabatrin both increase sedation. Use Caution/Monitor.

  • zaleplon

    levocetirizine and zaleplon both increase sedation. Use Caution/Monitor.

  • ziconotide

    levocetirizine and ziconotide both increase sedation. Use Caution/Monitor.

  • ziprasidone

    levocetirizine and ziprasidone both increase sedation. Use Caution/Monitor.

  • zolpidem

    levocetirizine and zolpidem both increase sedation. Use Caution/Monitor.

  • zonisamide

    levocetirizine and zonisamide both increase sedation. Use Caution/Monitor.

  • Xyzal (levocetirizine) dosing, indications, interactions, adverse effects, and more (2024)

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